Results for
""Receptors, Histamine H3""[mesh_terms]

Pitolisant (Wakix) for narcolepsy.

The Medical letter on drugs and therapeutics 2021;63(1617):19-21

Histamine H receptor ligands by hybrid virtual screening, docking, molecular dynamics simulations, and investigation of their biological effects.

Nakisa Ghamari, Omid Zarei, David Reiner, Siavoush Dastmalchi, Holger Stark, Maryam Hamzeh-Mivehroud

Chemical biology & drug design 2020;93(5):832-843

Assessment of receptor affinities of ophthalmic and systemic agents in dry eye disease.

Patrick Janeczko, Matthew R Norris, Leonard Bielory

Current opinion in allergy and clinical immunology 2021;21(5):480-485

Pharmacokinetic and pharmacodynamic assessment of histamine H receptor occupancy by enerisant: a human PET study with a novel H binding ligand, [C]TASP457.

Soichiro Kitamura, Yasuyuki Kimura, Keisuke Takahata, Toshiharu Shimazaki, Chie Seki, Yoko Ikoma, Masanori Ichise, Kazunori Kawamura, Makiko Yamada, Ming-Rong Zhang, Makoto Higuchi, Izumi Nishino, Tetsuya Suhara

European journal of nuclear medicine and molecular imaging 2022;49(4):1127-1135

Structure-based prediction of subtype selectivity of histamine H3 receptor selective antagonists in clinical trials.

Soo-Kyung Kim, Peter Fristrup, Ravinder Abrol, William A Goddard

Journal of chemical information and modeling 2012;51(12):3262-74

Modeling G protein-coupled receptors for structure-based drug discovery using low-frequency normal modes for refinement of homology models: application to H3 antagonists.

Brajesh K Rai, Gregory J Tawa, Alan H Katz, Christine Humblet

Proteins 2010;78(2):457-73

AZD5213: a novel histamine H3 receptor antagonist permitting high daytime and low nocturnal H3 receptor occupancy, a PET study in human subjects.

Aurelija Jucaite, Akihiro Takano, Emma Boström, Karl-Gustav Jostell, Per Stenkrona, Christer Halldin, Märta Segerdahl, Svante Nyberg

The international journal of neuropsychopharmacology 2014;16(6):1231-9

Sodium binding to hH3R and hH 4R--a molecular modeling study.

Andrea Strasser, Roland Seifert, Hans-Joachim Wittmann

Journal of molecular modeling 2015;20(8):2394