Filters

Clear all

Expert Opinion

Plain Language Summary

Expert Review

Text Availability

Abstract

Full text

Free full text

Publication Types

Journal Article

Research Support, Non-U.S. Gov't

Review

Randomized Controlled Trial

Comparative Study

Research Support, U.S. Gov't, P.H.S.

Clinical Trial

Research Support, N.I.H., Extramural

Multicenter Study

Publication Year

From

Quick links

Individual year

2024

2020

2017

2016

2014

2012

2009

2007

2004

Sort by:

selected

Print page

Email selected articles

Favourite selected articles

Create a NED Search Alert for this search

Save this search

Advanced Search

Run an advanced search

Results for
""Benzamidines""[mesh_terms]

12 Results

Searching titles within these results

Entropic cost of protein-ligand binding and its dependence on the entropy in solution.

Sheeba Jem Irudayam, Richard H Henchman

The journal of physical chemistry. B 2009;113(17):5871-84

Full Text

Abstract

Gibbs Free Energy of Hydrolytic Water Molecule in Acyl-Enzyme Intermediates of a Serine Protease: A Potential Application for Computer-Aided Discovery of Mechanism-Based Reversible Covalent Inhibitors.

Noriyuki Yamaotsu, Yosuke Masuda, Shuichi Hirono

Chemical & pharmaceutical bulletin 2017;65(10):889-892

Free Full Text

Abstract

Unusually strong binding to the DNA minor groove by a highly twisted benzimidazole diphenylether: induced fit and bound water.

Farial A Tanious, William Laine, Paul Peixoto, Christian Bailly, Kristie D Goodwin, Mark A Lewis, Eric C Long, Millie M Georgiadis, Richard R Tidwell, W David Wilson

Biochemistry 2007;46(23):6944-56

Free Full Text

Abstract

A computational simulation study of benzamidine derivatives binding to arginine-specific gingipain (HRgpA) from periodontopathogen Porphyromonas gingivalis.

Dooil Kim, Dae-Sil Lee

International journal of molecular sciences 2014;11(9):3252-65

Free Full Text

Abstract

DON/DRP-104 as potent serine protease inhibitors implicated in SARS-CoV-2 infection: Comparative binding modes with human TMPRSS2 and novel therapeutic approach.

Mahmoud E Soliman, Ernest Oduro-Kwateng

Journal of cellular biochemistry 2024;125(10):e30528

Full Text

Abstract

Preventive effect of trimidox on oxidative stress in U937 cell line.

Syu-Ichi Kanno, Mai Kakuta, Yasue Kitajima, Yuu Osanai, Kaori Kurauchi, Takaharu Ohtake, Mayuko Ujibe, Kouji Uwai, Mitsuhiro Takeshita, Masaaki Ishikawa

Biological & pharmaceutical bulletin 2007;30(5):994-8

Free Full Text

Abstract

Functional characterization of protein variants encoded by nonsynonymous single nucleotide polymorphisms in MARC1 and MARC2 in healthy Caucasians.

Gudrun Ott, Debora Reichmann, Cornelia Boerger, Ingolf Cascorbi, Florian Bittner, Ralf-Rainer Mendel, Thomas Kunze, Bernd Clement, Antje Havemeyer

Drug metabolism and disposition: the biological fate of chemicals 2014;42(4):718-25

Full Text

Abstract

A double-blind randomized controlled comparison of APDDR-0901, a novel cosmeceutical formulation, and 0.1% adapalene gel in the treatment of mild-to-moderate acne vulgaris.

Ha Eun Lee, Joo Yeon Ko, Young Hoon Kim, Seo Rye Yoo, Sang Ho Moon, Nack In Kim, Chun Wook Park, Jeong Hwan Kim, Hyun Ju Koh, Won Seok Park, Young Suck Ro

European journal of dermatology : EJD 2012;21(6):959-65

Full Text

Abstract

Unravelling high-affinity binding compounds towards transmembrane protease serine 2 enzyme in treating SARS-CoV-2 infection using molecular modelling and docking studies.

Pooja M, Gangavaram Jyothi Reddy, Kanipakam Hema, Sujatha Dodoala, Bharathi Koganti

European journal of pharmacology 2020;890():173688

Free Full Text

Abstract

Effect of NF-κB inhibition on chemoresistance in biliary-pancreatic cancer.

Katsuhiko Yanaga, Tadashi Uwagawa

Surgery today 2016;45(12):1481-8

Full Text

Abstract

Collagen degradation by host-derived enzymes during aging.

D H Pashley, F R Tay, C Yiu, M Hashimoto, L Breschi, R M Carvalho, S Ito

Journal of dental research 2004;83(3):216-21

Free Full Text

Abstract

Recent progress on inhibitors of the type II transmembrane serine proteases, hepsin, matriptase and matriptase-2.

Vishnu C Damalanka, James W Janetka

Future medicinal chemistry 2020;11(7):743-769

Full Text

Abstract

Results: 1 – 12 / 12

Filters

Expert Opinion

Text Availability

Publication Types

Publication Year

Results for ""Benzamidines""[mesh_terms]

Entropic cost of protein-ligand binding and its dependence on the entropy in solution.

Gibbs Free Energy of Hydrolytic Water Molecule in Acyl-Enzyme Intermediates of a Serine Protease: A Potential Application for Computer-Aided Discovery of Mechanism-Based Reversible Covalent Inhibitors.

Unusually strong binding to the DNA minor groove by a highly twisted benzimidazole diphenylether: induced fit and bound water.

A computational simulation study of benzamidine derivatives binding to arginine-specific gingipain (HRgpA) from periodontopathogen Porphyromonas gingivalis.

DON/DRP-104 as potent serine protease inhibitors implicated in SARS-CoV-2 infection: Comparative binding modes with human TMPRSS2 and novel therapeutic approach.

Preventive effect of trimidox on oxidative stress in U937 cell line.

Functional characterization of protein variants encoded by nonsynonymous single nucleotide polymorphisms in MARC1 and MARC2 in healthy Caucasians.

A double-blind randomized controlled comparison of APDDR-0901, a novel cosmeceutical formulation, and 0.1% adapalene gel in the treatment of mild-to-moderate acne vulgaris.

Unravelling high-affinity binding compounds towards transmembrane protease serine 2 enzyme in treating SARS-CoV-2 infection using molecular modelling and docking studies.

Effect of NF-κB inhibition on chemoresistance in biliary-pancreatic cancer.

Collagen degradation by host-derived enzymes during aging.

Recent progress on inhibitors of the type II transmembrane serine proteases, hepsin, matriptase and matriptase-2.

Results for
""Benzamidines""[mesh_terms]