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Caroline Schad, Ulrike Baum, Benjamin Frank, Uwe Dietzel, Felix Mattern, Carlos Gomes, Alicia Ponte-Sucre, Heidrun Moll, Uta Schurigt, Tanja Schirmeister

Antimicrobial agents and chemotherapy 2016;60(2):797-805

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Some physicochemical properties of the antitumor drug thiotepa and its metabolite tepa as obtained by density functional theory (DFT) calculations.

Djaffar Kheffache, Ourida Ouamerali

Journal of molecular modeling 2010;16(8):1383-90

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New cis-configured aziridine-2-carboxylates as aspartic acid protease inhibitors.

Christian Büchold, Yasmin Hemberger, Cornelia Heindl, Armin Welker, Björn Degel, Thomas Pfeuffer, Peter Staib, Sabrina Schneider, Philip J Rosenthal, Jiri Gut, Joachim Morschhäuser, Gerhard Bringmann, Tanja Schirmeister

ChemMedChem 2011;6(1):141-52

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The Inhibition of Cysteine Proteases Rhodesain and TbCatB: A Valuable Approach to Treat Human African Trypanosomiasis.

Maria Zappalà, Silvana Grasso, Gregorio Cullia, Lucia Tamborini, Santo Previti, Roberta Ettari

Mini reviews in medicinal chemistry 2017;16(17):1374-1391

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Metal Ion Complexes with Pyrazoles, Aziridines and Diaziridines - Synthesis and Biological Activity.

Paulina Mucha, Beata Sadowska, Ingo-Peter Lorenz, Katarzyna Malinowska

Current medicinal chemistry 2019;26(4):648-663

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Results for ""Aziridines""[mesh_terms]

Rational Tuning of the Reactivity of Three-Membered Heterocycle Ring Openings via S 2 Reactions.

Recent Developments in the Biosynthesis of Aziridines.

Synthesis of peptide macrocycles using unprotected amino aldehydes.

Cyclopropanation and aziridination catalyzed by non-heme iron and 2-oxoglutarate dependent enzymes.

EO-9 bladder instillations: formulation selection based on stability characteristics and in vitro simulation studies.

Enantiopure trans-3-arylaziridine-2-carboxamides: preparation by bacterial hydrolysis and ring-openings toward enantiopure, unnatural D-α-amino acids.

Anticancer drug-induced kidney disorders.

A discussion of the pH-dependent protonation behaviors of poly(2-(dimethylamino)ethyl methacrylate) (PDMAEMA) and poly(ethylenimine-ran-2-ethyl-2-oxazoline) (P(EI-r-EOz)).

Novel synthesis of 3,4-diaminobutanenitriles and 4-amino-2-butenenitriles from 2-(cyanomethyl)aziridines through intermediate aziridinium salts: an experimental and theoretical approach.

DNA Labeling Using DNA Methyltransferases.

Development of a New Antileishmanial Aziridine-2,3-Dicarboxylate-Based Inhibitor with High Selectivity for Parasite Cysteine Proteases.

Some physicochemical properties of the antitumor drug thiotepa and its metabolite tepa as obtained by density functional theory (DFT) calculations.

New cis-configured aziridine-2-carboxylates as aspartic acid protease inhibitors.

The Inhibition of Cysteine Proteases Rhodesain and TbCatB: A Valuable Approach to Treat Human African Trypanosomiasis.

Metal Ion Complexes with Pyrazoles, Aziridines and Diaziridines - Synthesis and Biological Activity.

Results for
""Aziridines""[mesh_terms]